Synthesis of ageladine A and analogs thereof

Peter Karuso (Inventor), Sudhir Ramnathrao Shengule (Inventor)

Research output: PatentResearch

Abstract

The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RrfCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.
LanguageEnglish
Patent numberUS20110152313
IPCA61K 31/437
Priority date20/06/08
Publication statusPublished - 23 Jun 2011

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Condensation
Patents and inventions
Aldehydes
Ageladine A

Bibliographical note

from CT/AU2009/000794

Cite this

Karuso, P., & Shengule, S. R. (2011). IPC No. A61K 31/437. Synthesis of ageladine A and analogs thereof. (Patent No. US20110152313).
Karuso, Peter (Inventor) ; Shengule, Sudhir Ramnathrao (Inventor). / Synthesis of ageladine A and analogs thereof. IPC No.: A61K 31/437. Patent No.: US20110152313.
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author = "Peter Karuso and Shengule, {Sudhir Ramnathrao}",
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Karuso, P & Shengule, SR 2011, Synthesis of ageladine A and analogs thereof, Patent No. US20110152313, IPC No. A61K 31/437.

Synthesis of ageladine A and analogs thereof. / Karuso, Peter (Inventor); Shengule, Sudhir Ramnathrao (Inventor).

IPC No.: A61K 31/437. Patent No.: US20110152313.

Research output: PatentResearch

TY - PAT

T1 - Synthesis of ageladine A and analogs thereof

AU - Karuso, Peter

AU - Shengule, Sudhir Ramnathrao

N1 - from CT/AU2009/000794

PY - 2011/6/23

Y1 - 2011/6/23

N2 - The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RrfCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

AB - The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RrfCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

UR - https://patentscope.wipo.int/search/en/detail.jsf?docId=US73278348

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Karuso P, Shengule SR, inventors. Synthesis of ageladine A and analogs thereof. A61K 31/437. 2011 Jun 23.