Synthesis of ageladine A and analogs thereof

Peter Karuso; Sudhir Ramnathrao Shengule

Synthesis of ageladine A and analogs thereof

Peter Karuso (Inventor), Sudhir Ramnathrao Shengule (Inventor)

Research output: Patent

Abstract

The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RrfCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

Original language	English
Patent number	US20110152313
IPC	A61K 31/437,C07D 471/02,A61P 35/00,A61P 27/02
Priority date	20/06/08
Filing date	19/06/09
Publication status	Accepted/In press - 23 Jun 2011

Bibliographical note

from CT/AU2009/000794

Cite this

@misc{46c19d52e511496a8dbecd7f5a3cee2d,

title = "Synthesis of ageladine A and analogs thereof",

abstract = "The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RrfCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.",

author = "Peter Karuso and Shengule, {Sudhir Ramnathrao}",

note = "from CT/AU2009/000794; US20110152313; A61K 31/437,C07D 471/02,A61P 35/00,A61P 27/02",

year = "2011",

month = jun,

day = "23",

language = "English",

type = "Patent",

}

TY - PAT

T1 - Synthesis of ageladine A and analogs thereof

AU - Karuso, Peter

AU - Shengule, Sudhir Ramnathrao

N1 - from CT/AU2009/000794

PY - 2011/6/23

Y1 - 2011/6/23

N2 - The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RrfCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

AB - The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RrfCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

UR - https://patentscope.wipo.int/search/en/detail.jsf?docId=US73278348

M3 - Patent

M1 - US20110152313

Y2 - 2009/06/19

ER -

Synthesis of ageladine A and analogs thereof

Abstract

Bibliographical note

Other files and links

Fingerprint

Cite this