Synthesis of ageladine A and analogs thereof

Peter Helmuth Karuso; Sudhir Ramnathrao Shengule

Synthesis of ageladine A and analogs thereof

Peter Helmuth Karuso (Inventor), Sudhir Ramnathrao Shengule (Inventor)

Macquarie University

Research output: Patent

Abstract

The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure R^dCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

Original language	English
Patent number	US2011152313
IPC	C07D 471/ 02 A I
Priority date	19/06/09
Publication status	Published - 23 Jun 2011

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title = "Synthesis of ageladine A and analogs thereof",

abstract = "The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RdCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.",

author = "Karuso, {Peter Helmuth} and Shengule, {Sudhir Ramnathrao}",

year = "2011",

month = jun,

day = "23",

language = "English",

type = "Patent",

note = "US2011152313; C07D 471/ 02 A I",

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TY - PAT

T1 - Synthesis of ageladine A and analogs thereof

AU - Karuso, Peter Helmuth

AU - Shengule, Sudhir Ramnathrao

PY - 2011/6/23

Y1 - 2011/6/23

N2 - The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RdCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

AB - The invention describes a one pot process for synthesizing a compound of structure (I), or a tautomer thereof. A compound of structure (II), or a tautomer thereof, and an aldehyde of structure RdCHO are condensed to form a condensation product. The resulting condensation product is then oxidized in the same reaction mixture to produce the compound of structure (I) or a tautomer thereof.

M3 - Patent

M1 - US2011152313

ER -

Synthesis of ageladine A and analogs thereof

Abstract

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